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Amphetamine is known to inhibit monoamine oxidase, Whilst the flexibility of amphetamine and its metabolites to inhibit numerous P450 isozymes and various enzymes has not been sufficiently elucidated. In vitro experiments with human microsomes point out minor inhibition of CYP2D6 by amphetamine and small inhibition of CYP1A2, 2D6, and 3A4 by one or